Adrenergic beta-2 Receptor Agonists

Name
Adrenergic beta-2 Receptor Agonists
Accession Number
DBCAT003416 (DBCAT000554, DBCAT002650)
Description

Compounds bind to and activate ADRENERGIC BETA-2 RECEPTORS.

Drugs
Drug Drug Description
Bitolterol Used to dilate air passages in the lungs that have become narrowed as a result of disease or inflammation. It is used in the treatment of asthma and chronic obstructive...
Abediterol Abediterol has been used in trials studying the treatment of Asthma, Chronic Obstructive Pulmonary Disease (COPD), and Chronic Obstructive Pulmonary Disease (COPD) and Asthma.
Orciprenaline A beta-2 adrenergic agonist used to treat bronchospasm, asthma, and COPD.
Salmeterol A long-acting beta-2 adrenergic receptor agonist used to treat asthma and COPD.
Formoterol An inhaled long-acting beta2-adrenergic receptor agonist used as a bronchodilator in the management of asthma and COPD.
Salbutamol A beta-2 adrenergic receptor agonist used to treat asthma, bronchitis, COPD, as well as prevent exercise induced bronchospasms.
Arformoterol A beta-2 adrenergic agonist and bronchodilator used for long term, symptomatic treatment of reversible bronchoconstriction in patients with chronic obstructive pulmonary disease (COPD), including chronic bronchitis and emphysema.
Indacaterol An inhaled long-acting beta-2 adrenergic agonist used to relax bronchial smooth muscle and improve symptoms and airflow obstruction caused by Chronic Obstructive Pulmonary Disease (COPD) and moderate to severe asthma.
Olodaterol A long-acting beta2-adrenergic agonist used in the management of chronic obstructive pulmonary disease (COPD), including chronic bronchitis and/or emphysema.
Levosalbutamol A beta-2 adrenergic receptor agonist used to treat COPD and asthma.
Ritodrine An adrenergic beta agonist used to treat premature labor.
Terbutaline A beta-2 adrenergic agonist used as a bronchodilator and to prevent premature labor.
Epinephrine A hormone and neurotransmitter used to treat allergic reactions, to restore cardiac rhythm, and to control mucosal congestion, glaucoma, and asthma.
Isoprenaline A catecholamine non-selective beta-adrenergic agonist typically used to treat bradycardia and heart block.
Procaterol A beta-2 adrenergic receptor agonist and bronchodilator used for the treatment of asthma and chronic obstructive pulmonary disease (COPD).
Clenbuterol A decongestant and bronchodilator used in a variety of respiratory conditions.
Fenoterol A beta-2 adrenergic agonist and bronchodilator used for the symptomatic treatment of asthma.
Pirbuterol A beta-2 adrenergic agonist and bronchodilator used for the symptomatic treatment of asthma.
Norepinephrine 拟交感的用于控制血压ssure during various hypotensive states and as an adjunct treatment during cardiac arrest.
Bambuterol A long acting beta2-adrenoceptor agonist for the management of lung diseases associated with bronchospasm.
Droxidopa A medication used to treat symptomatic neurogenic orthostatic hypotension (nOH) caused by dopamine beta-hydroxylase deficiency, non-diabetic autonomic neuropathy and primary autonomic failure caused by conditions such as Parkinson's disease.
Arbutamine Used to elicit acute cardiovascular responses (cardiac stumulant), similar to those produced by exercise, in order to aid in diagnosing the presence or absence of coronary artery disease (CAD) in...
Dobutamine A beta-1 agonist used to treat cardiac decompensation in patients with organic heart disease or from cardiac surgery.
Dipivefrin A prodrug of epinephrine used in ophthalmic solutions to reduce intraocular pressure in chronic open-angle glaucoma.
Ephedra sinica root An alpha and beta-adrenergic agonist used for the management of respiratory conditions related to bronchial asthma, such as wheezing, shortness of breath, and tightness of chest.
Isoetharine For the treatment of asthma, wheezing, and chronic asthmatic bronchitis.
Phenylpropanolamine A sympathomimetic that was previously used in nasal decongestants and weight loss products, but has been withdrawn by the FDA due to safety risks and lack of efficacy.
Vilanterol A long-acting beta2-adrenergic agonist used in combination with other bronchodilators for the management of chronic obstructive pulmonary disease (COPD), including chronic bronchitis and/or emphysema.
Celiprolol A beta-blocker for the management of hypertension and angina pectoris.
Doxofylline A methylxanthine derivative used in chronic obstructive pulmonary disease, asthma, and bronchospasms.
Protokylol Protokylol is a β-adrenergic receptor agonist used as a bronchodilator in Europe and the United States.
Racepinephrine A bronchodilator used to treat intermittent asthma.
Etafedrine A beta-2 adrenoceptor agonist used to treat a cough associated with inflamed mucosa.
PF-00610355 PF-00610355 has been used in trials studying the treatment of Lung Disease, Moxifloxacin, Pulmonary Disease, Asthma, Bronchial, and Bronchial Diseases, among others.
Hexoprenaline Hexoprenaline is a stimulant of beta 2 adrenergic receptors. It is used as a bronchodilator, antiasthmatic, and tocolytic agent.
Batefenterol Batefenterol has been used in trials studying the treatment of Pulmonary Disease, Chronic Obstructive.
Drugs & Drug Targets
Drug Target Type
Bitolterol Beta-2 adrenergic receptor target
Orciprenaline Beta-2 adrenergic receptor target
Salmeterol Beta-2 adrenergic receptor target
Salmeterol Cytochrome P450 3A4 enzyme
Salmeterol Cytochrome P450 2C8 enzyme
Salmeterol Cytochrome P450 3A5 enzyme
Salmeterol Cytochrome P450 3A7 enzyme
Salmeterol Beta-1 adrenergic receptor target
Salmeterol Beta-3 adrenergic receptor target
Salmeterol Serum albumin carrier
Salmeterol alpha1-acid glycoprotein carrier
Salmeterol 溶质载体家庭22个成员1 transporter
Salmeterol 溶解te carrier family 22 member 2 transporter
Salmeterol 溶解te carrier family 22 member 3 transporter
Formoterol Beta-2 adrenergic receptor target
Formoterol Beta-1 adrenergic receptor target
Formoterol Beta-3 adrenergic receptor target
Formoterol Cytochrome P450 2D6 enzyme
Formoterol Cytochrome P450 2C19 enzyme
Formoterol Cytochrome P450 2C9 enzyme
Formoterol Cytochrome P450 2A6 enzyme
Formoterol UDP-glucuronosyltransferase 1A1 enzyme
Formoterol UDP-glucuronosyltransferase 1-8 enzyme
Formoterol UDP-glucuronosyltransferase 1-9 enzyme
Formoterol UDP-glucuronosyltransferase 2B7 enzyme
Formoterol UDP-glucuronosyltransferase 2B15 enzyme
Formoterol 溶质载体家庭22个成员1 transporter
Formoterol 溶解te carrier family 22 member 4 transporter
Formoterol 溶解te carrier family 22 member 5 transporter
Formoterol 溶解te carrier family 22 member 3 transporter
Formoterol Serum albumin carrier
Salbutamol Beta-2 adrenergic receptor target
Salbutamol Beta-1 adrenergic receptor target
Salbutamol Cytochrome P450 3A4 enzyme
Salbutamol Beta-3 adrenergic receptor target
Arformoterol Beta-2 adrenergic receptor target
Arformoterol Cytochrome P450 2D6 enzyme
Arformoterol Cytochrome P450 2C19 enzyme
Arformoterol Cytochrome P450 2A6 enzyme
Arformoterol Cytochrome P450 2C9 enzyme
Indacaterol Beta-2 adrenergic receptor target
Indacaterol Cytochrome P450 3A4 enzyme
Indacaterol UDP-glucuronosyltransferase 1-1 enzyme
Indacaterol P-glycoprotein 1 transporter
Olodaterol Beta-2 adrenergic receptor target
Olodaterol Cytochrome P450 2C9 enzyme
Olodaterol Cytochrome P450 2C8 enzyme
Levosalbutamol Beta-2 adrenergic receptor target
Levosalbutamol 溶解te carrier organic anion transporter family member 1B1 transporter
Levosalbutamol 溶解te carrier organic anion transporter family member 1B3 transporter
Ritodrine Beta-2 adrenergic receptor target
Ritodrine 6-phosphogluconate dehydrogenase, decarboxylating enzyme
Ritodrine Sulfotransferase 1A1 enzyme
Ritodrine Sulfotransferase 1A3/1A4 enzyme
Ritodrine Beta adrenergic receptor target
Ritodrine ATP-sensitive potassium channel target
Ritodrine Calcium transporting ATPases target
Ritodrine Calcium-activated potassium channel target
Ritodrine Myosin light chain kinase, smooth muscle target
Ritodrine Sulfotransferase 1C4 target
Ritodrine Sulfotransferase enzyme
Ritodrine Sulfotransferase 1C4 enzyme
Terbutaline Beta-2 adrenergic receptor target
Terbutaline Cholinesterase enzyme
Terbutaline Beta-3 adrenergic receptor target
Terbutaline Beta-1 adrenergic receptor target
Terbutaline Sulfotransferase enzyme
Terbutaline UDP-glucuronosyltransferases (UGTs) enzyme
Terbutaline 溶解te carrier family 22 member 5 transporter
Terbutaline 溶解te carrier family 22 member 2 transporter
Epinephrine Alpha-1A adrenergic receptor target
Epinephrine Beta-1 adrenergic receptor target
Epinephrine Beta-2 adrenergic receptor target
Epinephrine 溶解te carrier family 22 member 2 transporter
Epinephrine 溶质载体家庭22个成员1 transporter
Epinephrine Cytochrome P450 2C9 enzyme
Epinephrine Cytochrome P450 3A4 enzyme
Epinephrine Alpha-1B adrenergic receptor target
Epinephrine Alpha-1D adrenergic receptor target
Epinephrine Alpha-2A adrenergic receptor target
Epinephrine Alpha-2B adrenergic receptor target
Epinephrine Tumor necrosis factor target
Epinephrine Catechol O-methyltransferase enzyme
Epinephrine Monoamine oxidase enzyme
Isoprenaline Beta-1 adrenergic receptor target
Isoprenaline Beta-2 adrenergic receptor target
Isoprenaline Beta-3 adrenergic receptor target
Isoprenaline Cytochrome P450 1A1 enzyme
Isoprenaline Superoxide dismutase [Cu-Zn] target
Isoprenaline Cytochrome P450 1B1 enzyme
Isoprenaline Serum albumin carrier
Isoprenaline Catechol O-methyltransferase enzyme
Isoprenaline Cholinesterase enzyme
Procaterol Beta-2 adrenergic receptor target
Clenbuterol Beta-2 adrenergic receptor target
Clenbuterol Beta-nerve growth factor target
Clenbuterol Tumor necrosis factor target
Clenbuterol Beta-1 adrenergic receptor target
Clenbuterol Beta-3 adrenergic receptor target
Clenbuterol Cytochrome P450 1A1 enzyme
Fenoterol Beta-2 adrenergic receptor target
Fenoterol Beta-1 adrenergic receptor target
Fenoterol Beta-3 adrenergic receptor target
Pirbuterol Beta-2 adrenergic receptor target
Pirbuterol Beta-1 adrenergic receptor target
Norepinephrine Phenylalanine-4-hydroxylase target
Norepinephrine Alpha-1A adrenergic receptor target
Norepinephrine Alpha-1B adrenergic receptor target
Norepinephrine Alpha-1D adrenergic receptor target
Norepinephrine Alpha-2A adrenergic receptor target
Norepinephrine Alpha-2B adrenergic receptor target
Norepinephrine Alpha-2C adrenergic receptor target
Norepinephrine Beta-1 adrenergic receptor target
Norepinephrine Beta-2 adrenergic receptor target
Norepinephrine Beta-3 adrenergic receptor target
Norepinephrine 溶解te carrier family 22 member 2 transporter
Norepinephrine 溶解te carrier family 22 member 3 transporter
Norepinephrine 溶解te carrier family 22 member 5 transporter
Norepinephrine 溶质载体家庭22个成员1 transporter
Norepinephrine POU domain, class 5, transcription factor 1 transporter
Norepinephrine Sodium-dependent noradrenaline transporter transporter
Norepinephrine Synaptic vesicular amine transporter target
Norepinephrine Chromaffin granule amine transporter target
Bambuterol Beta-2 adrenergic receptor target
Bambuterol Cholinesterase enzyme
Bambuterol Cholinesterase target
Droxidopa Phenylalanine-4-hydroxylase target
Droxidopa Alpha-1A adrenergic receptor target
Droxidopa Alpha-1B adrenergic receptor target
Droxidopa Alpha-1D adrenergic receptor target
Droxidopa Alpha-2A adrenergic receptor target
Droxidopa Alpha-2B adrenergic receptor target
Droxidopa Alpha-2C adrenergic receptor target
Droxidopa Beta-1 adrenergic receptor target
Droxidopa Beta-2 adrenergic receptor target
Droxidopa Beta-3 adrenergic receptor target
Droxidopa Aromatic-L-amino-acid decarboxylase enzyme
Droxidopa Monocarboxylate transporter 10 transporter
Droxidopa Sodium-dependent noradrenaline transporter transporter
Arbutamine Beta-1 adrenergic receptor target
Arbutamine Beta-2 adrenergic receptor target
Arbutamine Beta-3 adrenergic receptor target
Dobutamine Beta-1 adrenergic receptor target
Dobutamine Catechol O-methyltransferase enzyme
Dobutamine Beta-2 adrenergic receptor target
Dobutamine Alpha-1 adrenergic receptors target
Dobutamine Estrogen receptor alpha target
Dipivefrin Alpha-2A adrenergic receptor target
Dipivefrin Cholinesterase target
Dipivefrin Beta-2 adrenergic receptor target
Dipivefrin Alpha-1A adrenergic receptor target
Dipivefrin Acetylcholinesterase target
Ephedra sinica root Sodium-dependent dopamine transporter target
Ephedra sinica root Synaptic vesicular amine transporter target
Ephedra sinica root Chromaffin granule amine transporter target
Ephedra sinica root Sodium-dependent noradrenaline transporter target
Ephedra sinica root Amine oxidase [flavin-containing] A target
Ephedra sinica root Amine oxidase [flavin-containing] B target
Ephedra sinica root Sodium-dependent serotonin transporter target
Ephedra sinica root Alpha-2A adrenergic receptor target
Ephedra sinica root Alpha-2B adrenergic receptor target
Ephedra sinica root Alpha-2C adrenergic receptor target
Ephedra sinica root Beta-1 adrenergic receptor target
Ephedra sinica root Beta-2 adrenergic receptor target
Ephedra sinica root Beta-3 adrenergic receptor target
Isoetharine Beta-1 adrenergic receptor target
Isoetharine Beta-2 adrenergic receptor target
Phenylpropanolamine Amine oxidase [flavin-containing] A enzyme
Phenylpropanolamine Dopamine D1 receptor target
Phenylpropanolamine Beta-1 adrenergic receptor target
Phenylpropanolamine Beta-2 adrenergic receptor target
Phenylpropanolamine Alpha-2 adrenergic receptors target
Vilanterol Cytochrome P450 3A4 enzyme
Vilanterol Beta-2 adrenergic receptor target
Celiprolol Beta-1 adrenergic receptor target
Celiprolol Beta-2 adrenergic receptor target
Celiprolol Beta-3 adrenergic receptor target
Celiprolol Alpha-2A adrenergic receptor target
Celiprolol Alpha-2B adrenergic receptor target
Celiprolol Alpha-2C adrenergic receptor target
Celiprolol Cytochrome P450 2D6 enzyme
Doxofylline Phosphodiesterase 2A, cGMP-stimulated target
Doxofylline Adenosine receptor A2a target
Doxofylline Beta-2 adrenergic receptor target
Doxofylline Cytochrome P450 1A2 enzyme
Protokylol Beta-2 adrenergic receptor target
Racepinephrine Alpha-1A adrenergic receptor target
Racepinephrine Alpha-1B adrenergic receptor target
Racepinephrine Alpha-2A adrenergic receptor target
Racepinephrine Alpha-2B adrenergic receptor target
Racepinephrine Alpha-2C adrenergic receptor target
Racepinephrine Beta-1 adrenergic receptor target
Racepinephrine Beta-2 adrenergic receptor target
Racepinephrine Alpha-1D adrenergic receptor target
Racepinephrine Beta-3 adrenergic receptor target
Etafedrine Beta-2 adrenergic receptor target