γ-氨基丁酸的抑制高亲和性synaptosomal吸收bicyclo-heptane导数。

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Kovacs我Maksay G,西蒙尼M

γ-氨基丁酸的抑制高亲和性synaptosomal吸收bicyclo-heptane导数。

Arzneimittelforschung。1989年3月,39 (3):295 - 7。

PubMed ID
2502985 (在PubMed
]
文摘

2-phenyl-2 EGYT 3886 (dia (-) - (dimethylamino-ethoxy) - 1 r - 1, 7日7-trimethyl-bicyclo [2.2.1。]heptane hemifumarate) exhibiting anxiolytic and anticonvulsant properties is inactive on various binding sites of the GABAA (gamma-aminobutyric acid A) receptor/chloride ionophore complex, but is an effective inhibitor of high-affinity synaptosomal 3H-GABA uptake.

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